| 英文名稱 | Teneligliptin hydrobromide ( MP-513 hydrobromide) |
|---|---|
| 中文名稱 | 氫溴酸替格列汀 |
| CAS號 | 906093-29-6 |
| 分子式 | C44H65Br5N12O2S2 |
| 分子量 | 1,257.72 |
| 外觀 | Off-white to light brown |
| 儲存條件 | Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
| 英文名稱 | Teneligliptin hydrobromide ( MP-513 hydrobromide) |
|---|---|
| 中文名稱 | 氫溴酸替格列汀 |
| CAS號 | 906093-29-6 |
| 分子式 | C44H65Br5N12O2S2 |
| 分子量 | 1,257.72 |
| 外觀 | Off-white to light brown |
| 儲存條件 | Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
Teneligliptin (Teneligliptin hydrobromide anhydrous) is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50 values of approximately 1 nM.